TABLE. Antiretrovirals With Long-Acting Potential: Illustrative Examples from Different Drug Classes
Drug ClassARV NameDevelopment PhaseCompany
Non-Nucleoside
Reverse Transcriptase Inhibitor
RilpivirinePhase III injectable (oral agent approved)Janssen
Integrase InhibitorCabotegravirPhase III injectableViiV
Nucleoside/Nucleotide
Reverse Transciptase
Inhibitor (NRTI)
EFdAPhase IMerck
Tenofovir alafenamide fumarate (TAF)Preclinical implant (oral agent approved)Gilead
GS-9131Preclinical/Phase IGilead
Capsid InhibitorGS-CA1PreclinicalGilead